James E. Audia
100Patents
17h-index
96Co-inventors
89Inventor score
Filing activity: Aug 10, 1992 → Jun 11, 2024
Most-cited inventions
| Patent | Title | Area | Cited by | Status |
|---|---|---|---|---|
| US5614523A | Compounds having effects on serotonin-related systems | Chemistry; Metallurgy | 65 | Expired |
| US5789402A | Compounds having effects on serotonin-related systems | Chemistry; Metallurgy | 54 | Expired |
| US6509331B1 | Deoxyamino acid compounds, pharmaceutical compositions comprising same, and methods for inhibiting &bgr;-amyloid peptide release and/or its synthesis by use of such compounds | Chemistry; Metallurgy | 47 | Expired |
| US5627196A | Compounds having effects on serotonin-related systems | Chemistry; Metallurgy | 45 | Expired |
| US5708008A | 5-Substituted-3-(1,2,3,6-tetrahydropyridin-4-yl)-and 3-(piperidin-4-yl)-1H-indoles: new 5-HT.sub.1F agonists | Emerging Cross-Sectional Technologies | 45 | Expired |
| US9249161B2 | Bromodomain inhibitors and uses thereof | Chemistry; Metallurgy | 44 | Active |
| US5521197A | 3-<1-alkylenearyl>-4-<1,2,3,6-tetrahydropyridinyl>-and 3-<1-alkylenearyl>-4-piperidinyl-1h-indoles: new 5-HT.sub.1F agonists | Human Necessities | 40 | Expired |
| US5521196A | 5-HT.sub.1F agonists for the treatment of migraine | Human Necessities | 35 | Expired |
| US6191166A | Methods and compounds for inhibiting .beta.-amyloid peptide release and/or its synthesis | Chemistry; Metallurgy | 32 | Expired |
| US7648983B2 | BACE inhibitors | Human Necessities | 32 | Active |
| US5698571A | 5-HT.sub.1F mediated inhibition of neurogenic meningeal extravasation: a method for the treatment of migraine | Human Necessities | 24 | Expired |
| US5631265A | 8-substituted tetrahydro-beta-carbolines | Human Necessities | 24 | Expired |
| US5760051A | Tetrahydro-beta-carbolines | Chemistry; Metallurgy | 23 | Expired |
| US6211235A | Compounds for inhibiting .beta.-amyloid peptide release and/or its synthesis | Chemistry; Metallurgy | 20 | Expired |
| US9469646B2 | Modulators of methyl modifying enzymes, compositions and uses thereof | Chemistry; Metallurgy | 19 | Active |
| US5550134A | Methods for inhibiting bone loss | Human Necessities | 17 | Expired |
| US6506782B1 | Heterocyclic compounds, pharmaceutical compositions comprising same, and methods for inhibiting &bgr;-amyloid peptide release and/or its synthesis by use of such compounds | Human Necessities | 17 | Expired |
| US5670514A | Compositions for inhibiting bone loss | Human Necessities | 17 | Expired |
| US5629007A | Method of preventing prostatic cancer development | Human Necessities | 14 | Expired |
| US9409865B2 | Modulators of methyl modifying enzymes, compositions and uses thereof | Chemistry; Metallurgy | 14 | Active |
| US5869691A | Aminoalkyl-indoles | Chemistry; Metallurgy | 14 | Expired |
| US5721252A | 5HT.sub.1F agonists for the treatment of migraine | Human Necessities | 14 | Expired |
| US5635197A | Treatment and prevention of prostatic cancer metastasis | Human Necessities | 13 | Expired |
| US5688807A | Method for treating 5HT.sub.2B receptor related conditions | Chemistry; Metallurgy | 12 | Expired |
| US6153652A | N-(aryl/heteroaryl/alkylacetyl) amino acid amides, pharmaceutical compositions comprising same, and methods for inhibiting .beta.-amyloid peptide release and/or its synthesis by use of such compounds | Human Necessities | 12 | Expired |
Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.