Inventor · Village of La Jolla, CA, US

Nicholas David Peter COSFORD

38Patents
10h-index
56Co-inventors
78Inventor score

Filing activity: Nov 10, 1994 → Jul 29, 2021

Most-cited inventions

PatentTitleAreaCited byStatus
US5852041A Substituted pyridines useful as modulators of acethylcholine receptors Chemistry; Metallurgy 125 Expired
US6632823B1 Substituted pyridine compounds useful as modulators of acetylcholine receptors Chemistry; Metallurgy 50 Expired
US5723477A Modulators of acetylcholine receptors Chemistry; Metallurgy 36 Expired
US5585388A Substituted pyridines useful as modulators of acetylcholine receptors Chemistry; Metallurgy 30 Expired
US5736560A Substituted pyridines useful as modulators of acetylcholine receptors Chemistry; Metallurgy 27 Expired
US5703100A Modulators of acetylcholine receptors Chemistry; Metallurgy 25 Expired
US5594011A Modulators of acetylcholine receptors Chemistry; Metallurgy 24 Expired
US6656957B1 Pyridine derivatives Chemistry; Metallurgy 21 Expired
US6194581A Substituted pyridines useful as modulators of acetylcholine receptors Chemistry; Metallurgy 21 Expired
US5705512A Modulators of acetylcholine receptors Chemistry; Metallurgy 10 Expired
US5677459A Methods for the preparation of modulators of acetylcholine receptors Chemistry; Metallurgy 9 Expired
US7544677B2 Inhibitors of Akt activity Human Necessities 9 Expired
US9546174B2 Inhibitor of apoptosis protein (IAP) antagonists Emerging Cross-Sectional Technologies 8 Active
US6774138B2 Thiazolyl(pyridyl)ethyne compounds Chemistry; Metallurgy 7 Expired
US5686473A Substituted pyridines useful as modulators of acetylcholine receptors Chemistry; Metallurgy 7 Expired
US7589068B2 Inhibitors of Akt activity Human Necessities 7 Active
US6956049B1 Methods of modulating processes mediated by excitatory amino acid receptors Human Necessities 6 Expired
US7569592B2 Heteroaryl substituted pyrazole modulators of metabotropic glutamate receptor-5 Chemistry; Metallurgy 5 Expired
US7253190B2 Heteroaryl substituted tetrazole modulators of metabotrophic glutamate receptor-5 Chemistry; Metallurgy 5 Expired
US10047119B2 Inhibitor of apoptosis protein (IAP) antagonists Emerging Cross-Sectional Technologies 4 Active
US7105548B2 Heteroaryl substituted triazole modulators of metabotropic glutamate receptor-5 Chemistry; Metallurgy 4 Expired
US7365074B2 Pyridazine, pyrimidine and pyrazine ethyne compounds Chemistry; Metallurgy 3 Expired
US10544188B2 Inhibitor of apoptosis protein (IAP) antagonists Emerging Cross-Sectional Technologies 3 Active
US10300074B2 Use of inhibitor of apoptosis protein (IAP) antagonists in HIV therapy Human Necessities 3 Active
US7268151B2 Di-aryl substituted triazole modulators of metabotropic glutamate receptor-5 Chemistry; Metallurgy 3 Expired

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.