Patent · US Active

Pharmaceutical formulations of a bruton's tyrosine kinase inhibitor

US10010507B1 · kind B1 · utility

16Cited by
93References
28Claims
0Family size

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Key dates

Filing dateMar 1, 2018
Grant dateJul 3, 2018
Priority date
Expiry dateMar 1, 2038

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Described herein are pharmaceutical formulations of Bruton's tyrosine kinase (Btk) inhibitor 1-((R)-3-(4-amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one. Also disclosed are methods of using the Btk inhibitor, alone or in combination with other therapeutic agents, for the treatment of autoimmune diseases or conditions, heteroimmune diseases or conditions, cancer, including lymphoma, and inflammatory diseases or conditions.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.