Patent · US Active

Urea compounds and their use as enzyme inhibitors

US10023541B2 · kind B2 · utility

3Cited by
6References
8Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 19, 2016
Grant dateJul 17, 2018
Priority date
Expiry dateDec 19, 2036

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D233/88
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A compound having the following structure: or a pharmaceutically acceptable salt or derivative thereof. The compound may be used in the treatment or prevention of a disorder selected from appetite regulation, obesity, metabolic disorders, cachexia, anorexia, pain, inflammation, neurotoxicity, neurotrauma, stroke, multiple sclerosis, spinal cord injury, Parkinson's disease, levodopa-induced dyskinesia, Huntington's disease, Gilles de la Tourette's syndrome, tardive dyskinesia, dystonia, amyotrophic lateral sclerosis, Alzheimer's disease, epilepsy, schizophrenia, anxiety, depression, insomnia, nausea, emesis, alcohol disorders, drug addictions such as opiates, nicotine, cocaine, alcohol and psychostimulants, hypertension, circulatory shock, myocardial reperfusion injury, atherosclerosis, asthma, glaucoma, retinopathy, cancer, inflammatory bowel disease, acute and chronic liver disease such as hepatitis and liver cirrhosis, arthritis and osteoporosis.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.