Patent · US Active

Azabicyclo derivatives, process for preparation thereof and medical use thereof

US10085983B2 · kind B2 · utility

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Inventors

Yunzhou Jin · Shanghai, CN
Ping Bu · Shanghai, CN
Qi He · Zhuqiao, CN
Jiong Lan · Moraga, US
Fusheng ZHOU · Shanghai, CN
Liang Zhang · Sichuan, CN
Xiangyu He · Zhuqiao, CN

Key dates

Filing date	Sep 24, 2015
Grant date	Oct 2, 2018
Priority date	—
Expiry date	Sep 24, 2035

Classification

Technology area (CPC C)Chemistry; Metallurgy
CPC primaryC07D519/00
WIPO fieldPharmaceuticals
WIPO sectorChemistry

Abstract

Azabicyclo derivatives, a preparation process, and medical use thereof are provided. In particular, azabicyclo derivatives of formula (I), pharmaceutically acceptable salts, stereoisomers, solvates and prodrugs thereof are described. The azabicyclo derivatives of formula (I) are useful as Epidermal Growth Factor Receptor (EGFR) inhibitors. The definitions of the variable R groups in the azabicyclo derivatives of formula (I) are described in the specification.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.