Patent · US Active

Reversibly crosslinked micelle systems

US10106650B2 · kind B2 · utility

5Cited by
0References
1Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 14, 2012
Grant dateOct 23, 2018
Priority date
Expiry dateMay 14, 2032

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY10T428/2982
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides amphiphilic telodendrimers that aggregate to form nanocarriers characterized by a hydrophobic core and a hydrophilic exterior. The nanocarrier core may include amphiphilic functionality such as cholic acid or cholic acid derivatives, and the exterior may include branched or linear poly(ethylene glycol) segments. Nanocarrier cargo such as hydrophobic drugs and other materials may be sequester in the core via non-covalent means or may be covalently bound to the telodendrimer building blocks. Telodendrimer structure may be tailored to alter loading properties, interactions with materials such as biological membranes, and other characteristics.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.