Patent · US Active

11,13-modified saxitoxins for the treatment of pain

US10112953B2 · kind B2 · utility

3Cited by
4References
32Claims
0Family size

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Key dates

Filing dateSep 30, 2016
Grant dateOct 30, 2018
Priority date
Expiry dateSep 30, 2036

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Provided herein are compounds, pharmaceutical compositions comprising the compounds, methods of preparing the compounds, and methods of using the compounds and compositions in treating conditions associated with voltage-gated sodium channel function where the compounds are 11,13-modified saxitoxins according to Formula (I): where R1, X1 and X3 are as described herein.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.