Process for preparing ixazomib citrate and intermediates therefor
US10118937B1 · kind B1 · utility
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11Claims
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Key dates
| Filing date | Jan 3, 2018 |
| Grant date | Nov 6, 2018 |
| Priority date | — |
| Expiry date | Jan 3, 2038 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07F5/025
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
A process for making ixazomib citrate of formula VI comprising reacting a compound of formula V with citric acid to form ixazomib citrate of formula VI:
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.