Patent · US Active

Substituted pyrazolo[1,5-a]pyridine compounds as RET kinase inhibitors

US10174027B2 · kind B2 · utility

12Cited by
77References
30Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 29, 2017
Grant dateJan 8, 2019
Priority date
Expiry dateDec 29, 2037

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D519/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Provided herein are compounds of the General Formula I: and stereoisomers and pharmaceutically acceptable salts or solvates thereof, in which A, B, D, E, X1, X2, X3 and X4 have the meanings given in the specification, which are inhibitors of RET kinase and are useful in the treatment and prevention of diseases which can be treated with a RET kinase inhibitor, including diseases or disorders mediated by a RET kinase.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.