Patent · US Active

Fused pyrazole derivative having autotaxin inhibitory activity

US10189843B2 · kind B2 · utility

3Cited by
1References
11Claims
0Family size

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Key dates

Filing dateFeb 26, 2015
Grant dateJan 29, 2019
Priority date
Expiry dateFeb 26, 2035

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D519/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides a compound of formula (1), wherein R1, R2, R3, R4a, R4b, R5a and R5b are as defined in the description, which has an autotaxin inhibitory activity, a pharmaceutical composition comprising the compound as an active ingredient, and a method of prevention or treatment of a disease involving autotaxin, which is characterized by administering the compound.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.