Patent · US Active

Process for the preparation of Apixaban and intermediates thereof

US10208036B2 · kind B2 · utility

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5Claims
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Assignee

Inventors

Key dates

Filing dateSep 6, 2017
Grant dateFeb 19, 2019
Priority date
Expiry dateSep 6, 2037

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D211/86
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention refers to novel process for the preparation of Apixaban. Further, the invention also related to a process for the preparation of intermediate of Apixaban from very basic and cheap row material i.e. Aniline which is widely commercially available. The present invention provides process for preparation of Apixaban using a different sequence of synthetic steps and does not involve use of Ullmann reaction.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.