Patent · US Active

Pharmaceutical formulations of a Bruton's tyrosine kinase inhibitor

US10213386B2 · kind B2 · utility

11Cited by
95References
23Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 3, 2018
Grant dateFeb 26, 2019
Priority date
Expiry dateMay 3, 2038

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Described herein are pharmaceutical formulations of Bruton's tyrosine kinase (Btk) inhibitor 1-((R)-3-(4-amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one. Also disclosed are methods of using the Btk inhibitor, alone or in combination with other therapeutic agents, for the treatment of autoimmune diseases or conditions, heteroimmune diseases or conditions, cancer, including lymphoma, and inflammatory diseases or conditions.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.