Fungicidal N-cycloalkyl-N-{[ortho-(1-substituted-cycloalkyl)heteroaryl]methyl}(thio)carboxamides

US10244756B2 · kind B2 · utility

Assignee

• BAYER CROPSCIENCE AKTIENGESELLSCHAFT · DE

Inventors

• Pierre Cristau · Lyon, FR
• Philippe Desbordes · Val-de-Reuil, FR
• Julie GEIST · Val-de-Reuil, FR
• Lionel NICOLAS · Val-de-Reuil, FR
• Philippe Rinolfi · Villefranche-sur-Saône, FR
• Jan-Peter Schmidt · Folsom, US
• Tomoki Tsuchiya · Düsseldorf, DE

Key dates

• Filing date: May 19, 2016
• Grant date: Apr 2, 2019
• Expiry date: May 19, 2036

Classification

• Technology area (CPC C): Chemistry; Metallurgy
• CPC primary: C07D409/12
• WIPO field: Organic fine chemistry
• WIPO sector: Chemistry

Abstract

The invention relates to fungicidal N-cycloalkyl-N-{[ortho-(1-substituted-cycloalkyl)heteroaryl]methyl}carboxamides and their thiocarbonyl analogs of formula (I), their process of preparation, their use as fungicides, particularly in the form of fungicidal compositions, and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions. A represents a carbo-linked, unsaturated or partially saturated, optionally substituted 5-membered heterocyclyl group; T represents O or S; Z1 represents an optionally substituted C3-C7-cycloalkyl; p represents 1-5; B1 represents a carbo-linked, unsaturated, monocyclic or fused bicyclic 5-, 6-, 8-, 9-, 10-membered heterocyclyl ring, wherein the dotted line between the two adjacent carbons represents a single bond, a double bond or an aromatic bond.