Patent · US Active

Alvocidib prodrugs having increased bioavailability

US10259835B2 · kind B2 · utility

16Cited by
36References
13Claims
0Family size

Assignee

Inventors

Key dates

Filing dateAug 9, 2017
Grant dateApr 16, 2019
Priority date
Expiry dateAug 9, 2037

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D405/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds having the following structure (I): or a stereoisomer, tautomer or pharmaceutically acceptable salt thereof, wherein one of R1, R2 or R3 is —P(═O)(OH)2, and the other two of R1, R2 and R3 are each H, are provided. Pharmaceutical compositions comprising the compounds, and methods for use of the compounds for treating diseases associated with overexpression of a cyclin-dependent kinase (CDK) are also provided.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.