Patent · US Active

Diaryl macrocycle polymorph

US10294242B2 · kind B2 · utility

16Cited by
4References
20Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 5, 2016
Grant dateMay 21, 2019
Priority date
Expiry dateJul 5, 2036

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02P20/55
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

This disclosure relates to polymorphs of (7S,13R)-11-fluoro-7,13-dimethyl-6,7,13,14-tetrahydro-1,15-ethenopyrazolo[4,3-f][1,4,8,10]benzoxatriazacyclotridecin-4(5H)-one that are useful in the treatment of disease, such as cancer, in mammals. This disclosure also relates to compositions including such polymorphs, and to methods of using such compositions in the treatment of diseases, such as cancer, in mammals, especially in humans.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.