Patent · US Active

Derivatives of 3-heteroarylisoxazol-5-carboxylic amide useful for the treatment of inter alia cystic fibrosis

US10344023B2 · kind B2 · utility

6Cited by
11References
20Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 23, 2015
Grant dateJul 9, 2019
Priority date
Expiry dateDec 23, 2035

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D417/12
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present disclosure is based, in part, on the discovery that disclosed compounds can increase cystic fibrosis transmembrane conductance regulator (CFTR) activity as measured in human bronchial epithelial (hBE) cells.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.