Cyclic vinylogous amides as bromodomain inhibitors
US10351511B2 · kind B2 · utility
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4References
18Claims
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Key dates
| Filing date | Dec 14, 2017 |
| Grant date | Jul 16, 2019 |
| Priority date | — |
| Expiry date | Dec 14, 2037 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D295/21
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
Cyclic vinylogous amides of Formula I are disclosed The compounds are useful for treating diseases that arise from inappropriate activity of proteins containing an acetyl-lysine. The compositions comprise a genus of cyclic vinylogous amides that are inhibitors of bromodomain.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.