Patent · US Active

Pyrrolotriazinones and imidazotriazinones as ubiquitin-specific protease 7 inhibitors

US10351571B2 · kind B2 · utility

15Cited by
65References
17Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 24, 2018
Grant dateJul 16, 2019
Priority date
Expiry dateMay 24, 2038

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention relates to inhibitors of USP7 inhibitors useful in the treatment of cancers, neurodegenerative diseases, immunological disorders, inflammatory disorders, cardiovascular diseases, ischemic diseases, viral infections and diseases, and bacterial infections and diseases, having the Formula: where R1, R2, R3, R4, R5, R5′, R6, X1, X2, m, and n are described herein.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.