Patent · US Active

Heterocyclic-substituted pyridinopyrimidinone derivative as CDK inhibitor and use thereof

US10351578B2 · kind B2 · utility

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5Claims
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Assignee

Inventors

Key dates

Filing dateOct 9, 2018
Grant dateJul 16, 2019
Priority date
Expiry dateOct 9, 2038

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D513/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention relates to a heterocyclic-substituted pyridinopyrimidinone derivative and the use thereof as a therapeutically effective cyclin-dependent kinase (CDK) inhibitor. In particular, the present invention relates to the use of a new heterocyclic-substitute pyridinopyrimidinone derivative as shown in formula (I) and a pharmaceutical composition thereof as a selective CDK4/6 inhibitor in preventing or treating diseases related to CDK4/6.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.