Patent · US Active

Thiourea derivatives as activators of RORα and pharmaceutical composition containing same

US10407388B2 · kind B2 · utility

1Cited by
3References
10Claims
0Family size

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Inventors

Key dates

Filing dateMay 23, 2012
Grant dateSep 10, 2019
Priority date
Expiry dateJan 7, 2037

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P29/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Provided is a compound activating RORα gene, particularly a JC1 compound containing CGP52608 thiazolidinedione as a lead substance, and a pharmaceutically acceptable salt thereof. The compound is a lipid accumulation inhibitor and applicable to the treatment of metabolic diseases or inflammatory diseases.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.