Patent · US Active

N-(pyridin-2-yl)-4-(thiazol-5-yl)pyrimidin-2-amine derivatives as therapeutic compounds

US10479785B2 · kind B2 · utility

0Cited by
5References
29Claims
0Family size

Assignee

Inventors

Key dates

Filing dateAug 4, 2016
Grant dateNov 19, 2019
Priority date
Expiry dateAug 4, 2036

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P35/02
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

A novel class of inhibitors of protein kinases that are useful in the treatment of cell proliferative diseases and conditions, and especially those characterised by over-expression of CDK4, CDK6 and/or cyclin D, including certain cancers of lung, breast, brain, central nervous system, colorectal cancer and leukaemias. The inhibitors have the general structure I:

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.