Patent · US Active

Emulsion formulations of aprepitant

US10500208B2 · kind B2 · utility

8Cited by
2References
17Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJan 5, 2017
Grant dateDec 10, 2019
Priority date
Expiry dateMay 20, 2037

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Disclosed herein are novel pharmaceutical formulations of aprepitant suitable for parenteral administration including intravenous administration. Also included are formulations including both aprepitant and dexamethasone sodium phosphate. The pharmaceutical formulations are stable oil-in-water emulsions for non-oral treatment of emesis and are particularly useful for treatment of subjects undergoing highly emetogenic cancer chemotherapy.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.