Patent · US Active

WDR5 inhibitors and modulators

US10501466B2 · kind B2 · utility

3Cited by
1References
20Claims
0Family size

Assignee

Inventors

Key dates

Filing dateSep 19, 2018
Grant dateDec 10, 2019
Priority date
Expiry dateSep 19, 2038

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P35/02
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Described are N-(6-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-2-yl)-2,3-dihydro-1H-inden-1-yl)benzamide and acetamide-containing compounds that inhibit WDR5 and associated protein-protein interactions, pharmaceutical compositions including the compounds, and methods of using the compounds and compositions for treating disorders and conditions in a subject.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.