Patent · US Active

Quinazolinones and azaquinazolinones as ubiquitin-specific protease 7 inhibitors

US10513507B2 · kind B2 · utility

8Cited by
69References
20Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 11, 2017
Grant dateDec 24, 2019
Priority date
Expiry dateDec 11, 2037

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present disclosure relates to inhibitors of USP7 inhibitors useful in the treatment of cancers, neurodegenerative diseases, immunological disorders, inflammatory disorders, cardiovascular diseases, ischemic diseases, viral infections and diseases, and bacterial infections and diseases, having the Formula: where R1, R2, R3, R4, R4′, X1, Y1, Y2, Y3, Y4, n, and m are described herein.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.