Patent · US Active

Quinazolinones and azaquinazolinones as ubiquitin-specific protease 7 inhibitors

US10519130B2 · kind B2 · utility

8Cited by
69References
21Claims
0Family size

Assignee

Inventors

Key dates

Filing dateNov 2, 2018
Grant dateDec 31, 2019
Priority date
Expiry dateNov 2, 2038

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present disclosure relates to inhibitors of USP7 inhibitors useful in the treatment of cancers, neurodegenerative diseases, immunological disorders, inflammatory disorders, cardiovascular diseases, ischemic diseases, viral infections and diseases, and bacterial infections and diseases, having the Formula: where R1, R2, R3, R4, R4′, X1, Y1, Y2, Y3, Y4, n, and m are described herein.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.