Patent · US Active

Heterocyclic compounds useful in the treatment of disease

US10526298B2 · kind B2 · utility

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17References
47Claims
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Assignee

Inventors

Key dates

Filing dateJun 18, 2018
Grant dateJan 7, 2020
Priority date
Expiry dateJun 18, 2038

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D413/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Heterocyclic compounds are described that are lysophosphatidic acid receptor ligands that are useful in the treatment of lysophosphatidic acid receptor-dependent diseases and conditions, including but not limited to diseases involving fibrosis, such as fibrosis of the heart, kidney, liver and lung, and scleroderma; inflammatory diseases such as diabetic nephropathy and nonalcoholic steatohepatitis (NASH); ocular diseases such as diseases involving retinal degeneration; nerve diseases such as pruritus and pain.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.