Patent · US Active

Substituted pyrazole compounds as serine protease inhibitors

US10532995B2 · kind B2 · utility

0Cited by
24References
37Claims
0Family size

Assignee

Inventors

Key dates

Filing dateFeb 29, 2016
Grant dateJan 14, 2020
Priority date
Expiry dateFeb 29, 2036

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D417/14
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

There are provided inter alia multisubstituted aromatic compounds useful for the inhibition of thrombin and/or kallikrein, which compounds include substituted pyrazolyl. There are additionally provided pharmaceutical compositions. There are additionally provided methods of treating and preventing certain diseases or disorders, which diseases or disorders are amenable to treatment or prevention by the inhibition of thrombin and/or kallikrein.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.