Patent · US Active

Alpha-amino esters of hydroxypropylthiazolidine carboxamide derivative and salt form, crystal polymorph thereof

US10555934B2 · kind B2 · utility

2Cited by
5References
60Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJan 4, 2017
Grant dateFeb 11, 2020
Priority date
Expiry dateJan 4, 2037

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K9/48
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention provides pharmaceutical compositions comprising a compound of formula (I) or (II) and an additional therapeutic agent Also provided is the HCI salt and crystalline form of the compound of formula (I). The compounds inhibit the prostaglandin F receptor (PGF2alpha) and thus useful in the treatment of disorders such as preterm labor at the early gestational stage.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.