Patent · US Active

Pharmaceutical composition comprising dutasteride and propylene glycol monolaurate and preparation method of the same

US10561619B2 · kind B2 · utility

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0References
7Claims
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Assignee

Inventors

Key dates

Filing dateDec 29, 2016
Grant dateFeb 18, 2020
Priority date
Expiry dateDec 29, 2036

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to a pharmaceutical composition comprising dutasteride and propylene glycol monolaurate, which improves the stability of dutasteride, which is a poorly soluble drug as a 5-alpha reductase inhibitor, and a process for its preparation. More particularly, the present invention also relates to a capsule formulation which is smaller in size than a commercial dutasteride capsule formulation (AVODART®), but has the equivalent dissolution rate by preparing a pharmaceutical composition comprising propylene glycol monolaurate and dutasteride, which can improve the stability of the dutasteride. A dutasteride formulation having enhanced patient's compliance and improved stability and a method for producing the same are provided.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.