Patent · US Active

Alvocidib prodrugs having increased bioavailability

US10562925B2 · kind B2 · utility

8Cited by
94References
20Claims
0Family size

Assignee

Inventors

Key dates

Filing dateFeb 19, 2019
Grant dateFeb 18, 2020
Priority date
Expiry dateFeb 19, 2039

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D405/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds having the following structure (I): or a stereoisomer, tautomer or pharmaceutically acceptable salt thereof, wherein one of R1, R2 or R3 is —P(═O)(OH)2, and the other two of R1, R2 and R3 are each H, are provided. Pharmaceutical compositions comprising the compounds, and methods for use of the compounds for treating diseases associated with overexpression of a cyclin-dependent kinase (CDK) are also provided.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.