Patent · US Active

Pharmaceutical composition for oral administration

US10583087B2 · kind B2 · utility

1Cited by
1References
8Claims
0Family size

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Key dates

Filing dateApr 27, 2016
Grant dateMar 10, 2020
Priority date
Expiry dateApr 27, 2036

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P13/10
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Disclosed is a pharmaceutical composition for oral administration, comprising 1-{5-[(5-{[(2R)-2-ethylpyrrolidin-1-yl]methyl}-4-[4-methoxy-3-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl)carbamoyl]pyrazin-2-yl}pyperidine-4-carboxylic acid, which is a compound having pH-dependent solubility, or a pharmaceutically acceptable salt thereof, and a cellulose derivative. In the pharmaceutical composition for oral administration, the solubility and absorbability of the drug are improved.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.