Patent · US Active

Podophyllotoxin derivative with 4-position nitrogen substitution and preparation method and application thereof

US10639295B2 · kind B2 · utility

0Cited by
1References
6Claims
0Family size

Assignee

Inventors

Key dates

Filing dateAug 2, 2016
Grant dateMay 5, 2020
Priority date
Expiry dateAug 2, 2036

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K31/573
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A compound represented by formula (I) or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable formulation prepared using the compound and the salt. The compound represented by formula (I) or the pharmaceutically acceptable salt exhibits significantly higher buildup and concentration in the lungs compared to other tissues, a longer dwell time in the lungs, and/or elevated pharmaceutical efficacy.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.