Patent · US Active

Compounds

US10640498B2 · kind B2 · utility

4Cited by
0References
17Claims
0Family size

Assignee

Inventors

Key dates

Filing dateFeb 16, 2017
Grant dateMay 5, 2020
Priority date
Expiry dateFeb 16, 2037

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/10
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention relates to novel compounds of formula (I) and methods for the manufacture of inhibitors of deubiquitylating enzymes (DUBs). In particular, the invention relates to the inhibition of ubiquitin C-terminal hydrolase 30 or ubiquitin specific peptidase 30 (USP30). The invention further relates to the use of DUB inhibitors in the treatment of conditions involving mitochondrial dysfunction and in the treatment of cancer.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.