Patent · US Active

Composition and method for detecting hypoxia

US10695446B2 · kind B2 · utility

0Cited by
0References
17Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 2, 2016
Grant dateJun 30, 2020
Priority date
Expiry dateMay 2, 2036

Classification

  • Technology area (CPC G)Physics
  • CPC primaryG01N2800/7038
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A compound and method for detecting hypoxic cells and tissue are provided. The compound includes a probe selected from the group consisting of a hypoxia sensitive 2-nitroimidazole containing fluorescence imaging probe, a hypoxia sensitive reversible ON-OFF fluorescence imaging probe, a hypoxia sensitive azo-based fluorescence imaging probe, and combinations thereof. The method includes contacting the cells or tissue with the probe of any one of claims 1-13 and detecting fluorescent intensity of the cell or tissue, wherein increased fluorescent intensity indicates that the cells or tissue is hypoxic. Also provided are a method of synthesizing the compound and a method for synthesizing a therapeutic agent including the compound.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.