Substituted isoquinolines and phthalazines as rock kinase inhibitors
US10745381B2 · kind B2 · utility
0Cited by
2References
19Claims
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Assignee
Inventors
Key dates
| Filing date | Nov 6, 2019 |
| Grant date | Aug 18, 2020 |
| Priority date | — |
| Expiry date | Nov 6, 2039 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D471/04
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
The present invention relates to indoline-based compounds that inhibit Rho-associated protein kinase (ROCK) activity. In particular, the present invention relates to compounds, pharmaceutical compositions and methods of use, such as methods of inhibiting ROCK activity and methods for treating, for example cerebral cavernous malformation syndrome (CCM) and cardiovascular diseases using the compounds and pharmaceutical compositions of the present invention.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.