Patent · US Active

Enantiomers of the 1′,6′-isomer of neplanocin A

US10787478B2 · kind B2 · utility

0Cited by
12References
17Claims
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Assignee

Inventors

Key dates

Filing dateMar 8, 2019
Grant dateSep 29, 2020
Priority date
Expiry dateMar 8, 2039

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D473/34
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Enantiomers of 1′,6′-isoneplanocin, including derivatives of the enantiomers of 1′,6′-isoneplanocin, are disclosed along with novel synthetic methods. In particular, a substituted cyclopentane epoxide is synthesized into the enantiomers of 1′,6′-isoneplanocin. Enantiomers of carbocyclic nucleoside analogs of 3-deazaneplanocin to provide D- and L-like 1′,6′-iso-3-deazaneplanocin are also disclosed. The small molecule chemotherapeutic compounds beneficially provide DNA and RNA antiviral activity, demonstrating activity towards, for example, human cytomegalovirus, measles, Ebola, norovirus, dengue, vaccinia and HBV. Compounds exhibiting reduced S-adenosylhomocysteine hydrolase inhibitory effects are disclosed and provide improved toxicity profiles in comparison to neplanocin. The invention provides improved prophylactic and/or therapeutic antiviral efficacy.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.