Patent · US Active

Pharmaceutical formulations of a Bruton's tyrosine kinase inhibitor

US10828259B2 · kind B2 · utility

1Cited by
104References
25Claims
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Key dates

Filing dateApr 10, 2020
Grant dateNov 10, 2020
Priority date
Expiry dateApr 10, 2040

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Described herein are pharmaceutical formulations of Bruton's tyrosine kinase (Btk) inhibitor 1-((R)-3-(4-amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one. Also disclosed are methods of using the Btk inhibitor, alone or in combination with other therapeutic agents, for the treatment of autoimmune diseases or conditions, heteroimmune diseases or conditions, cancer, including lymphoma, and inflammatory diseases or conditions.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.