Patent · US Active

Stable amorphous form of sacubitril valsartan trisodium complex and processes for preparation thereof

US10857132B2 · kind B2 · utility

0Cited by
2References
23Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 10, 2017
Grant dateDec 8, 2020
Priority date
Expiry dateOct 10, 2037

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07B2200/13
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to stable amorphous form of sacubitril valsartan trisodium complex and its solid dispersion compounds, processes for their preparation and pharmaceutical composition comprising the same. The present invention also relates to an improved process for the preparation of sacubitril sodium and its use in the preparation of sacubitril valsartan trisodium complex.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.