Patent · US Active

Long-acting insulin or insulin analogue conjugate

US10894089B2 · kind B2 · utility

17Cited by
2References
15Claims
0Family size

Assignee

Inventors

Key dates

Filing dateFeb 17, 2016
Grant dateJan 19, 2021
Priority date
Expiry dateApr 12, 2036

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC12N2840/203
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to insulin and/or an insulin analogue conjugate, and a use thereof, wherein the insulin and/or insulin analogue have improved in vivo durability and stability by linking the same with an Fc region of immunoglobulin. The insulin and/or an insulin analogue conjugate of the present invention show an in vivo activity similar to that of insulin. In addition, the insulin and/or insulin analogue conjugate of the present invention are long-acting formulations of insulin and/or the analogue thereof, in which serum half-life is remarkably increased, and therefore, the present invention provides remarkable insulin and/or an insulin analogue conjugate, which do not induce hypoglycemia, a drawback of insulin treatment.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.