Patent · US Active

Thienopyrimidinones as ubiquitin-specific protease 7 inhibitors

US10906916B2 · kind B2 · utility

3Cited by
76References
16Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 18, 2019
Grant dateFeb 2, 2021
Priority date
Expiry dateJul 18, 2039

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02A50/30
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The disclosure relates to inhibitors of USP7 inhibitors useful in the treatment of cancers, neurodegenerative diseases, immunological disorders, inflammatory disorders, cardiovascular diseases, ischemic diseases, viral infections and diseases, and bacterial infections and diseases, having the Formula: where R1, R2, R3, R5, R5′, X1, X2, n, and m are described herein.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.