Patent · US Active

Phosphoramidate nucleoside derivatives as anticancer agents

US10906929B2 · kind B2 · utility

2Cited by
9References
16Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 31, 2017
Grant dateFeb 2, 2021
Priority date
Expiry dateMay 31, 2037

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07H19/173
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

This invention relates to derivatives of cladribine of Formula (I). The compounds are phosphoramidate derivatives in which the phosphoramidate moiety is situated on the 3′-hydroxyl group of cladribine. The invention also relates to pharmaceutical formulations of the cladribine derivatives and their use in methods of treatment. The compounds are useful in the treatment of cancer.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.