Patent · US Active

Inhibitors of KEAP1-Nrf2 protein-protein interaction

US10947252B2 · kind B2 · utility

2Cited by
0References
1Claims
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Assignee

Inventors

Key dates

Filing dateAug 19, 2019
Grant dateMar 16, 2021
Priority date
Expiry dateAug 19, 2039

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D519/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Sultam compounds, pharmaceutical compositions containing them, methods of making them, and methods of using them including methods for treating disease states, disorders, and conditions associated with the KEAP1-Nrf2 interaction, such as inflammatory bowel disease, including Crohn's disease and ulcerative colitis.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.