Patent · US Active

Tyrosine amide derivatives as Rho-Kinase inhibitors

US10954236B2 · kind B2 · utility

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15Claims
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Assignee

Inventors

Key dates

Filing dateOct 18, 2019
Grant dateMar 23, 2021
Priority date
Expiry dateOct 18, 2039

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D519/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Bicyclic dihydropyrimidine-carboxamide compounds of formula I described herein inhibit Rho Kinase and may be used for the treatment of many disorders associated with ROCK enzymes mechanisms, such as pulmonary diseases including asthma, chronic obstructive pulmonary disease (COPD), idiopathic pulmonary fibrosis (IPF) and pulmonary arterial hypertension (PAH).

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.