Patent · US Active

Compositions and methods for modulating HEXM1 expression

US10959966B2 · kind B2 · utility

1Cited by
0References
4Claims
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Key dates

Filing dateJan 30, 2015
Grant dateMar 30, 2021
Priority date
Expiry dateAug 17, 2035

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K45/06
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The potency of a series of Hexamethylene bis-acetamide (HMBA) derivatives of formula I, that induce Hexamethylene bis-acetamide inducible protein 1 (HEXIM1) was determined in cancer cells. The method of inducing HEXIM1 expression and cell differentiation in cancer and HIV cells are disclosed. Optimization of HMBA analogs that are symmetrical and unsymmetrical are also discussed.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.