Patent · US Active

Substituted [1,2,4]triazolo[1,5-a]pyrazines as LSD1 inhibitors

US10968221B2 · kind B2 · utility

5Cited by
39References
10Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 3, 2019
Grant dateApr 6, 2021
Priority date
Expiry dateOct 3, 2039

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention is directed to [1,2,4]triazolo[1,5-a]pyridine and [1,2,4]triazolo[1,5-a]pyrazine derivatives of Formula IIa, or a pharmaceutically acceptable salt thereof, which are LSD1 inhibitors useful in the treatment of diseases such as cancer.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.