Small molecules inhibitors of RAD51
US10973819B2 · kind B2 · utility
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Key dates
| Filing date | Mar 2, 2017 |
| Grant date | Apr 13, 2021 |
| Priority date | — |
| Expiry date | Mar 2, 2037 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D487/04
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
Embodiments concern methods and small molecule compositions for selectively inhibiting RAD51-mediated D-loop formation while preserving RAD51's ability to form nucleoprotein filaments. The selective RAD51 D-loop formation activity inhibitors DNA repair while minimizing replication-associated toxicity in normal tissue.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.