Patent · US Active

Anti-liferative agents comprising substituted benzo[e]pyrido[1,2-a][1,4]diazepines

US10975074B2 · kind B2 · utility

0Cited by
26References
30Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 13, 2019
Grant dateApr 13, 2021
Priority date
Expiry dateJun 13, 2039

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P35/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention relates to compounds comprising a substituted pyrrolo-, indolino- or tetrahydroisoquinoline-benzodiazepines alkylating moiety linked via the A-ring to aromatic groups of formula (Ia), and to pharmaceutically acceptable salts thereof, which are useful as medicaments, in particular as anti-proliferative agents.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.