Patent · US Active

Fused bicyclic inhibitors of menin-MLL interaction

US10975100B2 · kind B2 · utility

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Assignee

Inventors

Key dates

Filing dateFeb 13, 2020
Grant dateApr 13, 2021
Priority date
Expiry dateFeb 13, 2040

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P35/02
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to pharmaceutical agents useful for therapy and/or prophylaxis in a mammal, and in particular to fused bicyclic compounds, pharmaceutical composition comprising such compounds, and their use as menin/MLL protein/protein interaction inhibitors, useful for treating diseases such as cancer, myelodysplastic syndrome (MDS) and diabetes.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.