Patent · US Active

Pyrrolotriazinones and imidazotriazinones as ubiquitin-specific protease 7 inhibitors

US10981915B2 · kind B2 · utility

3Cited by
76References
12Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 24, 2019
Grant dateApr 20, 2021
Priority date
Expiry dateJun 24, 2039

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention relates to inhibitors of USP7 inhibitors useful in the treatment of cancers, neurodegenerative diseases, immunological disorders, inflammatory disorders, cardiovascular diseases, ischemic diseases, viral infections and diseases, and bacterial infections and diseases, having the Formula: where R1, R2, R3, R4, R5, R5′, R6, X1, X2, m, and n are described herein.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.