Patent · US Active

Crystalline solvate forms of a pharmaceutical

US10995112B2 · kind B2 · utility

0Cited by
38References
8Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 10, 2019
Grant dateMay 4, 2021
Priority date
Expiry dateNov 7, 2039

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07B2200/13
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Described herein are solid state 17α-ethynylandrost-5-ene-3β,7β,17β-triol including amorphous and crystalline forms and specific polymorphic forms thereof, and use of solid state 17α-ethynylandrost-5-ene-3β,7β,17β-triol in treating numerous diseases and disorders, including hyperglycemic conditions, such as type 2 diabetes and metabolic syndrome, autoimmune conditions, such as rheumatoid arthritis, ulcerative colitis and type 1 diabetes, among other inflammation related conditions, and neurodegenerative conditions in subjects or human patients.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.